ECHC 2016

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Sunday July 3, 2016
14:00Registration
Session chair:
Prof. Romano ORRU
(VU UNIVERSITY AMSTERDAM, Amsterdam, The Netherlands)
16:15Opening Ceremony
Prof. Vinod SUBRAMANIAM
(VRIJE UNIVERSITEIT AMSTERDAM, Amsterdam, The Netherlands)
16:30Opening Lecture - PL01 - How Natural Products Can Inspire Chemical Biology and Drug Discovery
Prof. Herbert WALDMANN
(MAX PLANCK INSTITUTE OF MOLECULAR PHYSIOLOGY, Dortmund, Germany)
17:15Welcome drink - sponsored by MDPI
Monday July 4, 2016
Session chair:
Dr Eelco RUIJTER
(VU UNIVERSITY AMSTERDAM, Amsterdam, The Netherlands)
09:00IL01 - Fluorinated Imaging Materials
Prof. Tobias RITTER
(MAX-PLANCK-INSTITUT FÜR KOHLENFORSCHUNG, Mulheim, Germany)
09:35PL02 - Organocatalytic Asymmetric Synthesis of Heterocycles
Prof. Dieter ENDERS
(RWTH AACHEN, Aachen, Germany)
10:20IL02 - The Development of Ligand Systems for Separating Minor Actinides from Lanthanides for Nuclear Fuel Reprocessing
Prof. Laurence HARWOOD
(UNIVERSITY OF READING, Reading, United Kingdom)
10:55Coffee break and Exhibition
Session chair:
Prof. Henk HIEMSTRA
(UNIVERSITY OF AMSTERDAM, Amsterdam, The Netherlands)
11:25IL03 - Stereoselective Heterocycle Synthesis Coupling Multicomponent Reactions with Biocatalysis or Organocatalysis
Prof. Luca BANFI
(UNIVERSITY OF GENOA, Genova, Italy)
12:00IL04 - Metal Free Cllick Reactions For Glycoconjugate Modification
Prof. Geert-Jan BOONS
(THE UNIVERSITY OF GEORGIA, Athens, GA, United States)
12:35IL05 - Target Family-Centric Privileged Structures: a Rich Playground for Diverse Heterocyclic Chemotypes
Dr Gerhard MÜLLER
(MERCACHEM, Martinsried, Germany)
13:10Lunch, Exhibition and Poster Session 1 (odd numbers)
Session chair:
Prof. Laurence HARWOOD
(UNIVERSITY OF READING, Reading, United Kingdom)
14:40Elsevier presentation: Data-Driven Discovery: Deriving and Applying Actionable Information in Medicinal Chemistry
15:00IL06 - Ynamides: Remarkable Building Blocks for Heterocyclic Synthesis
Prof. Gwilherm EVANO
(ULB, Brussels, Belgium)
Heterocyclic Synthetic MethodologyHeterocyclic Synthetic MethodologyMedicinal Chemistry and Chemical Biology
Session chair:
Prof. Laurence HARWOOD
(UNIVERSITY OF READING, Reading, United Kingdom)
Session chair:
Prof. Luca BANFI
(UNIVERSITY OF GENOA, Genova, Italy)
Session chair:
Dr Alessia AMORE
(UBIQ, Amsterdam, The Netherlands)
15:35KL01 - Alpha-Functionalization of Amines as a Tool for the Synthesis of Heterocycles and Natural Products
Prof. Till OPATZ
(JOHANNES GUTENBERG-UNIVERSITY, Mainz, Germany)
KL02 - First-in-Class MCRs Coupled with Cascade Reactions for the Generation of Molecular Complexity
Prof. Christopher HULME
(UNIVERSITY OF ARIZONA, Tucson, United States)
KL03 - Biomimetic Natural Product Synthesis
Dr Andrew LAWRENCE
(UNIVERSITY OF EDINBURGH, Edinburgh, United Kingdom)
16:00OC01 - Poxim: A Novel N-Heterocyclic Carbene Equipped with Multifunctional Phosphine Oxide
Prof. Yoichi HOSHIMOTO
(FACULTY OF ENGINEERING, OSAKA UNIVERSITY, Suita, Osaka, Japan)
OC06 - Asymmetric Synthesis of Natural Tetrahydroisoquinolines and Tetrahydroprotoberberines
Dr Steen INGEMANN JORGENSEN
(UNIVERSITY OF AMSTERDAM, Amsterdam, The Netherlands)
OC11 - Pyrazoloquinolinones, Revisited GABAA Receptor Tool Compounds
Mr David Chan Bodin SIEBERT
(TU WIEN, Wien, Austria)
16:20OC02 - Efficient Approach to the Synthesis of 2,3-Substituted Furo[2,3-b]Pyridines
Mr Fernando FUMAGALLI
(UNIVERSITY OF SAO PAULO, Ribeirao Preto, Brazil)
OC07 - Synthesis of 3-Benzazepines by Metal-Free Oxidative C-H Bond Functionalization-Ring Expansion Tandem Reaction
Mr Andrea GINI
(WISSENSCHAFTSZENTRUM STRAUBING, Straubing, Germany)
OC12 - Exploring Tryptophan Synthase as a Herbicidal Mode of Action
Dr Matthew MCLACHLAN
(SYNGENTA, Bracknell, Berkshire, United Kingdom)
16:40Coffee break and Exhibition
17:10OC03 - Rapid Composition of Spiranoid Lactones: Access to Natural and Unexplored Frames
Dr Dmitry TSVELIKHOVSKY
(THE HEBREW UNIVERSITY OF JERUSALEM, Jerusalem, Israel)
OC08 - Combining Photochemistry and Catalysis: Rapid Access to SP3 - Rich Polyheterocycles from Simple Pyrroles
Ms Emma BLACKHAM
(UNIVERSITY OF BRISTOL, Bristol, United Kingdom)
OC13 - The Allylic Azide Rearrangement in Tandem with Huisgen Cycloaddition: Synthesis of Diverse Polyhydroxylated Nitrogen Containing Scaffolds
Ms Rekha CHADDA
(SCHOOL OF CHEMISTRY, NUI GALWAY, Galway, Ireland)
17:30OC04 - Nitrosoallenes: Reactivity and Applications to Heterocycles Synthesis
Dr Hiroki TANIMOTO
(NARA INSTITUTE OF SCIENCE AND TECHNOLOGY, Nara, Japan)
OC09 - Intramolecular Tsuji-Trost Cascade Cyclization as a Novel Synthetic Strategy Towards Muironolide A
Mr John BRAUN
(VRIJE UNIVERSITEIT AMSTERDAM, Amsterdam, The Netherlands)
OC14 - Synthesis and Potential Cytotoxic Activity of New Substituted Indazole Derivatives Bearing Pyrrole and 2-Pyrone
Mr Mohamed EL GHOZLANI
(UNIVERSTY SULTAN MY SLIMAN, Béni Mellal, Morocco)
17:50OC05 - Synthesis of Highly and Diversely Substituted Heterocycles from Alk-3-yn-1-ones (Propargyl Ketones)
Prof. Roman DEMBINSKI
(OAKLAND UNIVERSITY, Rochester, MI, United States)
OC10 - C-Brigded N-Heterocycles as New Ligands
Mr Tim-Daniel J. STUMPF
(JUSTUS-LIEBIG-UNIVERSITY GIESSEN, Giessen, Germany)
OC15 - Towards a Biomimetic Synthesis of Sciodole
Mr Josh HOMER
(UNIVERSITY OF AUCKLAND, Auckland, New Zealand)
18:10End of the day
Tuesday July 5, 2016
Session Chair:
Dr Tommi MEULEMANS
(MERCACHEM-SYNCOM, Nijmegen, The Netherlands)
09:00PL03 - Catalytic Approaches from the Synthesis of Enantiopure Biologically Relevant Heterocycles
Prof. Floris RUTJES
(RADBOUD UNIVERSITY NIJMEGEN, Nijmegen, The Netherlands)
09:45PL04 - Carbo- and Heterocycles via Metal-Catalyzed Cycloadditions
Dr Fernando LOPEZ
(UNIVERSITY OF SANTIAGO DE COMPOSTELA (USC) AND SPANISH NATIONAL RESEARCH COUNCIL (CSIC), Santiago de Compostela, Spain)
10:30IL07 - Photoactive Molecular and Supramolecular Materials Built-up with Heterocycles
Prof. Gianluca M. FARINOLA
(UNIVERSITY OF BARI, Bari, Italy)
11:05Coffee break and Exhibition
Session Chair:
Prof. Huib OVAA
(NETHERLANDS CANCER INSTITUTE, Leiden, The Netherlands)
11:30IL08 - Redesigning the Molecules of Nature: Lessons Learned from Total Synthesis
Prof. Karl GADEMANN
(UNIVERSITY OF ZÜRICH, Zürich, Switzerland)
12:05IL09 - Copper Catalysis for Synthesis of Enantiopure Alcohols, Amines and Heteroarenes
Prof. Syuzanna HARUTYUNYAN
(UNIVERSITY OF GRONINGEN, Groningen, The Netherlands)
12:40IL10 - C-H Functionalization for the Synthesis and Assembly of Heterocycles
Prof. Lutz ACKERMANN
(GEORG-AUGUST UNIVERSITY GOETTINGEN, Goettingen, Germany)
13:15Lunch, Exhibition and Poster Session 2 (even numbers)
Session Chair:
Prof. Hermen OVERKLEEFT
(LEIDEN UNIVERSITY, Leiden, The Netherlands)
14:45IL11 - Catalysis: A Versatile Tool for the Synthesis of Nitrogen-Containing Heterocycles
Dr Geraldine MASSON
(INSTITUT DE CHIMIE DES SUBSTANCES NATURELLES CNRS, Gif-sur-Yvette, France)
Heterocyclic Synthetic MethodologyHeterocyclic Synthetic MethodologyMedicinal Chemistry and Chemical Biology
Session Chair:
Prof. Hermen OVERKLEEFT
(LEIDEN UNIVERSITY, Leiden, The Netherlands)
Session Chair:
Prof. Lutz ACKERMANN
(GEORG-AUGUST UNIVERSITY GOETTINGEN, Goettingen, Germany)
Session Chair:
Prof. Henk TIMMERMAN
(VU UNIVERSITY AMSTERDAM, Oegstgeest, The Netherlands)
15:20KL04 - New Tricks for Old Heterocycles: from Natural Product Synthesis to Click-Like Functionalizations
Prof. Johan WINNE
(UGENT, Ghent, Belgium)
KL05 - Synthesis of New Spiroacetals by Sustainable Gold Catalysis
Prof. Norbert KRAUSE
(DORTMUND UNIVERSITY OF TECHNOLOGY, Dortmund, Germany)
KL06 - New Multicomponent Reactions and Strategies to Heterocyclic and Macrocyclic Peptides
Dr Daniel GARCÍA RIVERA
(LEIBNIZ INSTITUTE OF PLANT BIOCHEMISTRY / UNIVERSITY OF HAVANA, La Habana, Cuba)
15:45OC16 - Synthesis of Highly Enantioenriched Pyrrolo[1,2-a]Quinolines. Organocatalyzed Domino Cyclopropane Ring Opening/aza-Michael/aldol Reaction Followed by Acid-Promoted Lactamization
Mr Eduardo SANCHEZ
(UPV/EHU UNIVERSITY OF THE BASQUE COUNTRY, Leioa, Spain)
OC21 - Is Gold Catalysis a Competitive Method toward Heterocycles ?
Mrs Solène MIASKIEWICZ
(STRASBOURG UNIVERSITY, Strasbourg, France)
OC26 - Palladium-Catalyzed Isocyanide Insertion in Construction of Diverse Heterocycles
Dr Esther VICENTE GARCIA
(VRIJE UNIVERSITEIT AMSTERDAM, Amsterdam, The Netherlands)
16:05OC17 - Brönsted-Acid Catalysed C2-Alkenylation of Aromatic Nitrogen Heterocycles
Mr Giacomo CRISENZA
(UNIVERSITY OF BRISTOL, Bristol, United Kingdom)
OC22 - Aliphatic N-Heterocycle Synthesis through Direct C-H Bond Amination
Mr Petrus KUIJPERS
(UNIVERSITY OF AMSTERDAM, Amsterdam, The Netherlands)
OC27 - Biologically Active Indolines - Novel Multi-Functional Indolinic Drugs for the Treatment of Inflammatory Diseases
Prof. Abraham NUDELMAN
(BAR ILAN UNIVERSITY, Ramat Gan, Israel)
16:25Coffee break and Exhibition
17:00OC18 - Rearrangement and Cycloaddition Reactions of Donor-Acceptor Cyclopropanes
Prof. Daniel B. WERZ
(TU BRAUNSCHWEIG, Braunschweig, Germany)
OC23 - 3-Diazoindolin-2-Imines: A Novel Class of Metal Carbene Precursors for the Syntheses of Indole Derivatives
Prof. Yanguang WANG
(ZHEJIANG UNIVERSITY, Hangzhou, China)
OC28 - Asymmetric Reduction of Enamines towards the Synthesis of (-)-Cytisine and Heterocyclic Building Blocks
Mr Hugo REGO CAMPELLO
(UNIVERSITY OF BRISTOL, Bristol, United Kingdom)
17:20OC19 - Pd- and Cu-Catalyzed Stereo- and Regiocontrolled Decarboxylative / C-H Alkenylation of Heroarenes
OC24 - Donor-Acceptor Cyclopropanes in Synthesis of Azaheterocycles
Prof. Igor TRUSHKOV
(M V LOMONOSOV MOSCOW STATE UNIVERSITY, Moscow, Russia)
OC29 - Biology-Oriented Synthesis Based on Privileged Structures: Building Framework Diversity Around Pyrrole Cores
Prof. José Carlos MENÉNDEZ
(UNIVERSIDAD COMPLUTENSE, Madrid, Spain)
17:40OC20 - Enantioselective Organocatalyzed Α-Sulfanylation of Isoxazolidin-5-ones: An Approach To b2,2-Amino Acids
Mr Timothée CADART
(LABORATOIRE COBRA UMR 6014, ROUEN, France)
OC25 - Chirality in Boron-Chelated Dipyrromethene Fluorophores: Synthesis and Chiroptical Investigations
Dr Michael HALL
(NEWCASTLE UNIVERSITY, Newcastle upon Tyne, United Kingdom)
OC30 - Exploring the Antifungal and Antibiofilm Properties of Imidazolium Salts and Fluorescent Benzannulated Benzimidazoles
Prof. Henri SCHREKKER
(UNIVERSIDADE FEDERAL DO RIO GRANDE DO SUL, Porto Alegre-RS, Brazil)
18:00End of the day
18:30Boat tour and Conference dinner
Wednesday July 6, 2016
Session Chair:
Prof. Karl Anker JOERGENSEN
(AARHUS UNIVERSITY, Aarhus, Denmark)
09:00IL12 - Complex Natural Product as a Driving Force for Discovery in Organic Synthesis and Chemical Biology
Prof. Xiaoguang LEI
(PEKING UNIVERSITY, Beijing, China)
09:35IL13 - Metallation–Substitution of Saturated Nitrogen Heterocycles
Prof. Iain COLDHAM
(UNIVERSITY OF SHEFFIELD, Sheffield, United Kingdom)
10:10PL05 - Springer Junior Heterocyclic Chemistry Award Lecture (chaired by Bert Maes, editor of Springer)
Exploiting the Reactivity of Strained Rings and Hypervalent Bonds for the Synthesis of Heterocycles
Prof. Jerome WASER
(EPFL, Lausanne, Switzerland)
10:55IL14 - α-Perluoroalkylated Cyclic Imines as a Valuable Building Blocks
Prof. Dr Valentine G. NENAJDENKO
(MOSCOW STATE UNIVERSITY, Moscow, Russia)
11:30Coffee break and Exhibition
Session Chair:
Prof. Floris RUTJES
(RADBOUD UNIVERSITY NIJMEGEN, Nijmegen, The Netherlands)
11:55IL15 - New Strategies for the Synthesis of Heterocyclic through Multicomponent Reactions and Metal-Catalyzed Isomerization
Prof. Thomas NIELSEN
(NOVO NORDISK, Copenhagen N, Denmark)
12:30PL06 - Making Molecular Prosthetics with a Small Molecule Synthesizer
Prof. Martin D. BURKE
(UNIVERSITY OF ILLINOIS, Urbana, United States)
13:15Lunch
Heterocyclic Synthetic MethodologyEnabling TechnologiesMedicinal Chemistry and Chemical Biology
Session Chair:
Prof. Martin D. BURKE
(UNIVERSITY OF ILLINOIS, Urbana, United States)
Session Chair:
Dr Maikel WIJTMANS
(VU UNIVERSITY AMSTERDAM, Amsterdam, The Netherlands)
Session Chair:
Prof. Rob LEURS
(VU UNIVERSITY AMSTERDAM, Amsterdam, The Netherlands)
14:15KL07 - Gamma-Alkylidenebutenolides and Gamma-Hydroxybutyrolactams: Preparation and Reactivity
Dr Laurent COMMEIRAS
(AIX-MARSEILLE UNIVERSITY, Marseille cedex 20, France)
KL08 - Functionalization of Heterocycles via C–H Activation and Photoredox Catalysis in Batch and Continuous Flow
Dr Timothy NOEL
(EINDHOVEN UNIVERSITY OF TECHNOLOGY, Eindhoven, The Netherlands)
KL09 - Going Beyond ß-Amino Acid Derivatives as Inhibitors of Cathepsin A
Dr Sven RUF
(SANOFI-AVENTIS DEUTSCHLAND GMBH, Frankfurt am Main, Germany)
14:40OC31 - Picolinic Acid Ligand-Promoted Palladium-Catalyzed C-H Acetoxylation of Simple Arenes
Dr M. Angeles FERNANDEZ-IBANEZ
(UNIVERSITY OF AMSTERDAM, Amsterdam, The Netherlands)
OC36 - N-Heterocyclic Carbene Ligands in Iridium Complexes for the Detection of Pyridine Analogues in NMR by Non-Hydrogenative Para-Hydrogen Induced Hyperpolarization
Dr Martin FEITERS
(RADBOUD UNIVERSITY, Nijmegen, The Netherlands)
OC41 - Designing Residence Time into Heterocyclic Ligands for Drug Targets
Dr Julien LOUVEL
(LACDR, Leiden, The Netherlands)
15:00OC32 - Stereoselective Transformations of 2h-Chromene Derivatives
Prof. Tibor KURTÁN
(UNIVERSITY OF DEBRECEN, Debrecen, Hungary)
OC37 - Expansion of the Concept of Nonlinear Effects in Catalytic Reactions Beyond Asymmetric Catalysis
Prof. Michael SCHNÜRCH
(TU WIEN, Wien, Austria)
OC42 - Photopharmacology
Mr Mickel HANSEN
(RIJKSUNIVERSITEIT GRONINGEN, Groningen, The Netherlands)
15:20Coffee break and Exhibition
15:50OC33 - Scope and Limitations of the Organocatalyzed Domino Vinylogous Aldol Oxa Michael Reaction
Ms Larissa GEIGER
(KARLSRUHE INSTITUTE OF TECHNOLOGY, Karlsruhe, Germany)
OC38 - Direct Heteroatom Incorporating Ester to Arene Transformation: Modular Synthesis of Fluorescent Dyes
Mr Christian FISCHER
(UNIVERSITY OF BASEL, Basel, Switzerland)
OC43 - Novel Synthesis of Tetrahydroisoquinoline Derivatives Using Petasis Reaction
Dr Agnieszka GRAJEWSKA
(ADAM MICKIEWICZ UNIVERSITY, Poznan, Poland)
16:10OC34 - Dearomative Arylation of Electrophilic Indoles for the Total Synthesis of Natural Products
Prof. Guillaume VINCENT
(UNIVERSITÉ PARIS SUD INSTITUT DE CHIMIE MOLÉCULAIRE ET DES MATÉRIAUX D'ORSAY (ICMMO), Orsay, France)
OC39 - Methodology Development Towards the Lasso Peptide Series
Prof. Jan VAN MAARSEVEEN
(UNIVERSITEIT VAN AMSTERDAM, Amsterdam, The Netherlands)
OC44 - Palladium Catalyzed C-Arylation of Amino Acid Derived Hydantoins
Mr Josep MAS ROSELLO
(UNIVERSITY OF BRISTOL, Bristol, United Kingdom)
16:30OC35 - Integrative Methodology for Iterative Theory-Experiment Driven Multicomponent Reaction Development
Mr Art KRUITHOF
(VU AMSTERDAM, Amsterdam, The Netherlands)
OC40 - A Lab-Scale Reactor for the Continuous Generation of Anhydrous Diazomethane
Dr Doris DALLINGER
(UNIVERSITY OF GRAZ, Graz, Austria)
OC45 - Enantioselective Synthesis of 4-Arylpyridine Atropisomers by Central-to-Axial Chirality Conversion
Ms Ophélie QUINONERO
(ISM2 - INSTITUT DES SCIENCES MOLÉCULAIRE DE MARSEILLE, Marseille, France)
Session Chair:
Prof. Romano ORRU
(VU UNIVERSITY AMSTERDAM, Amsterdam, The Netherlands)
16:50PL07 - Organocatalysis for Diversity-Oriented Synthesis
Prof. Karl Anker JOERGENSEN
(AARHUS UNIVERSITY, Aarhus, Denmark)
17:35Poster prizes
Prof. Romano ORRU
(VU UNIVERSITY AMSTERDAM, Amsterdam, The Netherlands)
17:50End of the Symposium

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