12th EFMC Short Course on Medicinal Chemistry
Sunday April 24, 2016
18:00Dinner
20:00Opening
20:15Basic Principles of Enzymology
Dr Laurie LEBRUN
(CELGENE, San Diego, United States)
Monday April 25, 2016
07:30Breakfast
08:30Introduction
09:00Protein Kinase Inhibitors
Dr Gerhard MÜLLER
(MERCACHEM, Martinsried, Germany)
10:30Coffee Break
11:00Epigenetic Target Families in Medicinal Chemistry
Prof. Paul BRENNAN
(UNIVERSITY OF OXFORD, Oxford, United Kingdom)
12:30Lunch
13:30BETting on Epigenetic Targets: From Phenotypic Discovery to First Time in Man
Dr Chun-wa CHUNG
(GLAXOSMITHKLINE R&D, Stevenage, United Kingdom)
15:00Coffee Break
15:30Hands on Tutorial - Case Study I: Development of a Kinase Inhibitor
Dr Leon VAN BERKOM (MERCACHEM-SYNCOM, Nijmegen, The Netherlands)
Dr Toine VAN DEN BERGH (MERCACHEM-SYNCOM, Nijmegen, The Netherlands)
18:00Day End
Tuesday April 26, 2016
07:30Breakfast
08:30Proteases as Drug Targets
Dr Holger SELLNER
(NOVARTIS PHARMA AG, Basel, Switzerland)
10:00Coffee Break
10:30Proteasome Inhibitors
Prof. Michael GROLL
(TECHNISCHE UNIVERSITÄT MÜNCHEN, Garching, Germany)
12:00Lunch
13:00Glycomimetics - an Underexplored Compound Class for Medicinal Chemistry
Prof. Dr Beat ERNST
(UNIVERSITY OF BASEL, Basel, Switzerland)
14:30Coffee Break
15:00Hands on Tutorial - Case Study II: Development of a HIV Medicine
Dr Stijn GREMMEN (MERCACHEM, Nijmegen, The Netherlands)
Dr Harald ALBERS (MERCACHEM-SYNCOM, Nijmegen, The Netherlands)
17:30Day End
Wednesday April 27, 2016
07:30Breakfast
08:30The PDE Family and Inhibitors
Dr Andrew BELL
(IMPERIAL COLLEGE LONDON, London, United Kingdom)
10:00Coffee break
10:30Fragment-Based Lead Generation
Prof. Iwan DE ESCH
(VRIJE UNIVERSITEIT AMSTERDAM, Amsterdam, The Netherlands)
12:30Wrap-up and Lunch

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