13th EFMC Short Course on Medicinal Chemistry
Sunday April 23, 2017
17:00Registration
18:00Dinner
Monday April 24, 2017
07:30Breakfast
08:30Introduction
09:00Mathematics of binding kinetics
Prof. Georges VAUQUELIN
(VUB, Brussel, Belgium)
10:30Coffee Break
11:00Mathematics of binding kinetics - Part II
Prof. Georges VAUQUELIN
(VUB, Brussel, Belgium)
12:30Lunch
13:30Characterizing the Dynamics of Molecular Interactions
Prof. Helena DANIELSON
(UPPSALA UNIVERSITY, Uppsala, Sweden)
15:00Coffee Break
15:30Characterizing the Dynamics of Molecular Interactions - Part II
Prof. Helena DANIELSON
(UPPSALA UNIVERSITY, Uppsala, Sweden)
17:00Day End
18:00Dinner and walking tour through Leiden
Tuesday April 25, 2017
07:30Breakfast
08:30Kinetics for drug discovery: In vitro assays to study GPCRs
Dr Laura HEITMAN
(UNIVERSITY OF LEIDEN, Leiden, The Netherlands)
10:00Coffee Break
10:30Kinetics in Drug Discovery - A Case for G Protein-coupled Receptors
Prof. Ad P. IJZERMAN
(UNIVERSITY OF LEIDEN, Leiden, The Netherlands)
12:00Lunch
13:00Pharmacokinetic-pharmacodynamic Relationships, the Connecting Role of Binding Kinetics
Dr Liesbeth DE LANGE (UNIVERSITY OF LEIDEN, Leiden, The Netherlands)
Mr Wilbert DE WITTE (UNIVERSITY OF LEIDEN, Leiden, The Netherlands)
15:00Coffee Break
15:30Pharmacokinetic-pharmacodynamic Relationships, the Connecting Role of Binding Kinetics - Part II
Mr Wilbert DE WITTE (UNIVERSITY OF LEIDEN, Leiden, The Netherlands)
Dr Liesbeth DE LANGE (UNIVERSITY OF LEIDEN, Leiden, The Netherlands)
17:00Day End
18:00Dinner
Wednesday April 26, 2017
07:30Breakfast
08:30The Use of Kinetic Data in Early Drug Discovery: HSP90 as a Model to Gain Mechanistic Insight into Drug Binding Kinetics
Dr Matthias FRECH
(MERCK, Darmstadt, Germany)
10:00Coffee Break
10:30The Use of Kinetic Data in Early Drug Discovery: HSP90 as a Model to Gain Mechanistic Insight into Drug Binding Kinetics - Part II
Dr Matthias FRECH
(MERCK, Darmstadt, Germany)
12:00Wrap-up and Lunch

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