XVI International Conference on Heterocycles in Bioorganic Chemistry
Metz, France June 8-11, 2015
Session Chair:
Opening
PL01 - Photoreactive Heterocycles and Natural Product Derivatives
Coffee Break
Session Chair:
PL02 - Targeting DNA Methylation: a Medicinal Chemistry Approach
IL01 - Synthetic Explorations in Small-ring Azaheterocyclic Chemistry and Development of Novel Bioactive Heterocycles
OC01 - Heterocycle-Peptide Hybrids: Synthesis, Conformational Analysis, and Utilization in Medicinal Chemistry
Lunch
Session Chair:
PL03 - The Importance of Heterocycles in Agrochemistry: Fungicides as a Case Study
IL02 - Synthesis of Biorelevant Heterocycles with N-heterocyclic Carbenes
OC02 - Exploiting the Zincke Reaction to Produce Sophisticated Heptamethine Dyes
OC03 - Diverse Synthesis of Natural Product Inspired Fused and Spiro-Heterocyclic Scaffolds via Ring Distortion And Construction Strategy
OC04 - Novel Cross-Conjugated Dienones Based on 4-Piperidone Moiety: Synthesis and Antitumor Properties
Coffee Break and Poster Session 1
Welcome Reception (in the Exhibition area)
Session Chair:
PL04 - Non Noble Metal Catalysis for Making Precious Molecules
IL03 - Synthesis of Novel Alpha7-nAchR Ligands: from an Idea to in Rodent Results for Alzheimer [18F] TEP Imaging
OC05 - Recent Advances in the Total Synthesis of Phormidolides B and C
Coffee Break
Session Chair:
PL05 - Metal Catalysis for Heteroarene Synthesis
IL04 - New Methods in Thioamide Chemistry
Lunch
Session Chair:
PL06 - The Discovery and Development of the HIV Intergrase Inhibitors Dolutegravir and Cabotegravir
IL05 - Are Generic Drugs Only a Copy_and_Paste Products?
OC06 - An Original Domino Radical Cyclisation/Smiles Rearrangement Combination: Application to the Synthesis of Indolo[2,3-b]Quinoline-Type Derivatives
OC07 - Palladium-Catalyzed Cross-Coupling Reactions in the Asymmetric Synthesis of Pyrrolo[1,2-b]Isoquinolines
OC08 - Synthesis of Long Regioregular Dialkyl-Substituted Alpha-Oligofurans
Coffee Break and Poster Session 2
Session chair:
PL07 - Bronsted Acid and Metal-catalyzed Reactions in the Synthesis of Heterocycles
IL06 - Utilization of Hypervalent Iodonium Reagents for the Construction and Functionalization of Heterocyclic Molecules
OC09 - Synthesis of Agrochemistry-Related F-Heterocycles from Novel Fluorinated Diazoalkanes
Coffee Break
OC10 - Flavylium-Based Pigments – “Click” Synthesis & Biological Relevance
OC11 - Synthesis of 7-(2-Aminophenyl)- and 7-(4-Aminophenyl)Guanine, DNA Adducts Derived from the Phenylnitrenium Ion
OC12 - Heterocyclic Coumarine Analogs as Zinc Metalloprotease Inhibitors
Lunch
Session chair:
IL07 - Silicon-Containing Tetrahydrocyclopenta[C]Acridine Derivatives as CDKs Inhibitors: Design, Organometallic Synthesis, Metabolic Stability And Optimization
OC13 - Synthesis of Imidazo-Pyrrolo-Pyrazines/Diazepines/Diazocines via Domino Ugi/Micheal Reaction and Silver-Catalyzed Heteroannulation
OC14 - Synthesis and Antifungal Activity of N-Acyl Derivatives of 1,4-Benzoxazin- and 1,4-Benzoxazepin-3-ONES
OC15 - Mixed Cu(II) Cu(I) Complexes with Bioheterocycles as the Platform for Construction of Novel Anticancer Agents
Coffee Break
Excursions
Banquet
Session chair:
PL08 - Heterocycles Derived from Natural Products in Management of Multidrug Resistance
IL08 - At the Crossroads of Chemistry and Biology: Inhibiting Protein Kinase CK2 by Heterocyclic Small Molecules
Coffee Break
Session chair:
IL09 - Overcoming Resistance with beta-Lactams
OC16 - Discovery Of Novel Thieno[3,2-b]Pyrrole 5-Carboxamides as Potent Inhibitors of Chikungunya Virus (CHIKV)
Closing