Small Molecule Protein Degraders: A New Opportunity for Drug Design and Development
Oegstgeest (near Leiden), The Netherlands April 23-26, 2023
Registration
Dinner at the hotel
Get Together at the Castle Bar
Opening
Introduction to Small Molecule Degraders: PROTACS and Molecular Glues - Part 1
Coffee Break
Introduction to Small Molecule Degraders: PROTACS and Molecular Glues - Part 2
Lunch
The Ternary Complex E3-Degrader-Target: Biophysical Binding Assays and Structures - Part 1
Coffee Break
The Ternary Complex E3-Degrader-Target: Biophysical Binding Assays and Structures - Part 2
Day End
Walking tour through Leiden
Dinner in Leiden
The Current & Future Clinical Landscape of Molecular Degraders of Disease-Causing Proteins - Part 1
Coffee Break
The Current & Future Clinical Landscape of Molecular Degraders of Disease-Causing Proteins - Part 2
Lunch
Medicinal Chemistry Optimisation of Small Molecule Degraders - Part 1
Coffee Break
Medicinal Chemistry Optimisation of Small Molecule Degraders - Part 2
Day End
Dinner at the hotel
Get Together at the Castle Bar
Importance of Cellular Degradation Kinetics and Mechanisms for Development of Potent Therapeutic Degraders - Part 1
Coffee Break
Importance of Cellular Degradation Kinetics and Mechanisms for Development of Potent Therapeutic Degraders - Part 2
Wrap up and Lunch