16th EFMC Short Course on Medicinal Chemistry

New Opportunities in GPCR Drug Discovery

 Oegstgeest (near Leiden), The Netherlands    May 8-11, 2022

Confirmed Speakers

Discovery of H1/H4 Dual Ligands

Prof. Iwan DE ESCH
Prof. Iwan DE ESCH
VRIJE UNIVERSITEIT AMSTERDAM, Amsterdam, The Netherlands

GPCR Ligand Design: Cheminformatics and Modelling

Dr Chris DE GRAAF
Dr Chris DE GRAAF
SOSEI HEPTARES, Cambridge, United Kingdom
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GPCR Ligands: Molecular Recognition, Kinetics and Allosteric Modulation

Dr Laura HEITMAN
Dr Laura HEITMAN
UNIVERSITY OF LEIDEN, Leiden, The Netherlands
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Binding and Modulating GPCRs by Inside/Outside Binding Nanobodies

Dr Raimond HEUKERS
Dr Raimond HEUKERS
QVQ, Utrecht, The Netherlands
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Discovery of Cariprazine, A Dopamine D3 Receptor Prefering Third Generation Antipsychotics

Prof. Gyorgy KESERU
Prof. Gyorgy KESERU
HUNGARIAN ACADEMY OF SCIENCES, Budapest, Hungary
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A General Introduction into GPCRdb & Hands-on with the GPCRdb

Dr Albert KOOISTRA
Dr Albert KOOISTRA
UNIVERSITY OF COPENHAGEN, København, Denmark
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Partial Agonism/Biased Signalling and its Therapeutical Relevance

Dr Rob LANE
Dr Rob LANE
UNIVERSITY OF NOTTINGHAM, Nottingham, United Kingdom
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General Introduction to GPCRs: Pharma Relevance, Indications, Molecular Pharmacology

Prof. Rob LEURS
Prof. Rob LEURS
VRIJE UNIVERSITEIT AMSTERDAM, Amsterdam, The Netherlands
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System Biology Approaches to GPCR Targets

Dr Aurelien RIZK
Dr Aurelien RIZK
INTERAX BIOTECH, Villigen, Switzerland
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The ‘Hunger Games’ - Structural Studies of the MC4 Receptor Reveal Mechanism for Satiety

Dr Moran SHALEV-BENAMI
Dr Moran SHALEV-BENAMI
WEIZMANN INSTITUTE, Rehovot, Israel
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